Faculty Information - KITAMURA Masanori

Educational Background

Research Field (Keyword)

Work experience /Academic appointments

Publications

Invited Lectures

（Last updated : 2023-02-16 11:41:42）

KITAMURA Masanori
Department Matsuyama University School of Clinical Pharmacy, College of Pharmaceutical Sciences

Position Professor

Educational Background

2000/04～2003/03

〔Doctoral course〕, Graduate School, Division of Pharmaceutical Sciences, Hokkaido University, Completed,

Research Field (Keyword)

Organic chemistry, Synthetic chemistry, Chemical pharmacy, Bio-related chemistry (Key Word：Organic Chemistry, Bio-organic Chemistry, Bio-inorganic Chemistry)

Work experience /Academic appointments

1.	2003/04～2004/03	Kyoto University Department of Chemistry, Graduate School of Science Researcher
2.	2004/04～2007/03	Kyoto University Department of Chemistry, Graduate School of Science Special researcher of the Japan Society for the Promotion of Science
3.	2007/04～2011/11	Tokyo University of Science Faculty of Pharmaceutical Sciences Assistant Professor
4.	2011/11～2020/03	Kanazawa University Faculty of Pharmaceutical Sciences, Institute of Medical, Pharmaceutical, and Health Sciences Associate Professor

Publications

1.	2022/10	Article	Measurement of Hepatic CYP3A4 and 2D6 Activity Using Radioiodine-Labeled O-Desmethylvenlafaxine (Collaboration)
2.	2021/04	Article	Development of a triazinedione-based dehydrative condensing reagent containing 4-(dimethylamino)pyridine as an acyl transfer catalyst (Collaboration)
3.	2020/03	Article	Trizaine-based dehydrative condensation reagents bearing carbon-substituents (Collaboration)
4.	2019/12	Article	Development of Triazinone-Based Condensing Reagents for Amide Formation (Collaboration)
5.	2019/07	Article	Preparation of Alkyl Ethers with Diallyltriazinedione‐Type Alkylating Agents (ATTACKs-R) Under Acid Catalysis (Collaboration)
6.	2019/07	Article	Substitution of the Dimethylamino Group in Gramines and One-Pot Cyclization to Tetrahydro-β-carbolines Using a Triazine-Based Activating Agent (Collaboration)
7.	2018/06	Article	Imido-substituted triazines as dehydrative condensing reagents for the chemoselective formation of amides in the presence of free hydroxy groups (Collaboration)
8.	2018/04	Article	An isolable and bench-stable epoxidizing reagent based on triazine: Triazox (Collaboration)
9.	2018/02	Article	Development of highly electron-deficient and less sterically-hindered phosphine ligands possessing 1,3,5-triazinyl groups (Collaboration)
10.	2017	Article	Novel Alkylating Reagents Designed by the Characteristics of 1,3,5-Triazines (Collaboration)
11.	2017	Article	Study of O-Allylation using Triazine-based Reagents (Collaboration)
12.	2016	Article	Alcohol- and Amine-Tolerant Synthesis of Six-Membered Cyclic Quaternary Ammonium Salts by Using a Triazine-Based Reagent (Collaboration)
13.	2016	Article	Development of a Triazine-Based tert-Butylating Reagent, TriAT-tBu (Collaboration)
14.	2016	Article	Development of Acid-Catalyzed Fluorous Benzylating Reagents Based on a Triazinedione Core (Collaboration)
15.	2016	Article	Increased Plasma Concentrations of Unbound SN-38, the Active Metabolite of Irinotecan, in Cancer Patients with Severe Renal Failure (Collaboration)
16.	2016	Article	Potent triazine-based dehydrocondensing reagents substituted by an amido group (Collaboration)
17.	2015	Book	Supramolecular Hosts and Catalysts Formed by Synergitic Molecular Assemblies of Multinuclear Zinc(II) Complexes in Aqueous Solutions (Collaboration)
18.	2015	Article	O-Benzylation of Carboxylic Acids Using 2,4,6-Tris(benzyloxy)-1,3,5-triazine (TriBOT) under Acidic or Thermal Conditions (Collaboration)
19.	2015	Article	Radiogallium Complex-Conjugated Bifunctional Peptides for Detecting Primary Cancer and Bone Metastases Simultaneously (Collaboration)
20.	2014	Article	Design and Synthesis of Chiral Zn2+ Complexes Mimicking Natural Aldolases for Catalytic C–C Bond Forming Reactions in Aqueous Solution (Collaboration)
21.	2014	Article	Development of a New Benzylating Reagent Spontaneously Releasing Benzyl Cation Equivalents at Room Temperature (Collaboration)
22.	2014	Article	pecific Labeling of Streptavidin for Better Understanding of Ligand Modification in Modular Method for Affinity Labeling (MoAL) (Collaboration)
23.	2014	Article	Role of Linkers in Tertiary Amines That Mediate or Catalyze 1,3,5-Triazine-Based Amide-Forming Reactions (Collaboration)
24.	2014	Article	Synthesis of Pyrrolidinium Salts using a Triazine-based Reagent under Mild Conditions (Collaboration)
25.	2013	Book	4-(4,6-Dimethoxy-1,3,5-triazin-2-yl)-4-methylmorpholinium chloride. (Collaboration)
26.	2013	Article	A Practical Method for p-Methoxybenzylation of Hydroxy Groups Using 2,4,6-Tris(p-methoxybenzyloxy)-1,3,5-triazeine (TriBOT-PM) (Collaboration)
27.	2013	Article	Asymmetric Aldol Reactions between Acetone and Benzaldehydes Catalyzed by Chiral Zn2+ Complexes of Aminoacyl 1,4,7,10-Tetraazacyclododecane: Fine-Tuning of the Amino-Acid Side Chains and a Revised Reaction Mechanism (Collaboration)
28.	2013	Article	Binding of Sulforhodamine B to Human Serum Albumin: A Spectroscopic Study (Collaboration)
29.	2013	Article	Development and Evaluation of a Radiobromine-labeled Sigma Ligand for Tumor Imaging (Collaboration)
30.	2013	Article	Study of 1,3,5-triazine-based Catalytic Amide-forming Reactions: Effect of Solvents and Basicity of Reactants (Collaboration)
31.	2012	Article	Molecular Recognition of Hydrocarbon Guests by a Supramolecular Capsule Formed by the 4:4 Self-assembly of Tris(Zn2+–cyclen) and Trithiocyanurate in Aqueous Solution (Cyclen = 1,4,7,10-Tetraazacyclododecane) (Collaboration)
32.	2012	Article	One-Pot Chemoenzymatic Synthesis of Chiral 1,3-Diols Using an Enantioselective Aldol Reaction with Chiral Zn2+ Complex Catalysts and Enzymatic Reduction Using Oxidoreductases with Cofactor Regeneration (Collaboration)
33.	2011	Article	11B NMR Sensing of d-Block Metal Ions in Vitro and in Cells Based on the Carbon-Boron Bond Cleavage of Phenylboronic Acid-Pendant Cyclen (Cyclen = 1,4,7,10-Tetraazacyclododecane) (Collaboration)
34.	2011	Article	Design and Synthesis of Photocleavable Biotinylated-dopamine with Polyethyleneoxy Photocleavable Linkers (Collaboration)
35.	2011	Article	Photochemical Cleavage Reaction of 8-Quinolinyl Sulfonates That are Halogenated and Nitrated at the 7-Position (Collaboration)
36.	2011	Article	Regioselective Aromatic Substitution Reactions of Cyclometalated Ir(III) Complexes: Synthesis and Photochemical Properties of Substituted Ir(III) Complexes That Exhibit Blue, Green, and Red Color Luminescence Emission (Collaboration)
37.	2010	Article	Design and Synthesis of a Fluorescent Probe for Zn2+, 5,7-Bis(N,N-dimethylaminosulfonyl)-8-hydroxyquinoline-Pendant 1,4,7,10-Tetraazacyclododecane and Zn2+-Dependent Hydrolytic and Zn2+-Independent Photochemical Reactivation of Its Benzenesulfonyl-Caged Derivative (Collaboration)
38.	2010	Article	Molecular Recognition of Inositol 1,4,5-Trisphosphate and Model Compounds in Aqueous Solution by Ditopic Zn2+ Complexes Containing Chiral Linkers (Collaboration)
39.	2009	Article	Chiral Catalysts Dually Functionalized with Amino Acid and Zn2+ Complex Components for Enantioselective Direct Aldol Reactions Inspired by Natural Aldolases: Design, Synthesis, Complexation Properties, Catalytic Activities, and Mechanistic Study (Collaboration)
40.	2009	Article	Guidelines for Pattern Recognition using Differential Receptors and Indicator Displacement Assays (Collaboration)
41.	2008	Article	Combinatorial Approach for the Design of New, Simplified Chiral Phase-transfer Catalysts with High Catalytic Performance for Practical Asymmetric Synthesis of α-Alkyl-α-amino Acids (Collaboration)
42.	2008	Article	Combinatorial Design of Simplified High Performance Chiral Phase-transfer Catalysts for Practical Asymmetric Synthesis of α-Alkyl- and α,α-Dialkyl-α-amino Acids (Collaboration)
43.	2007	Article	New, Chiral Phase Transfer Catalysts for Effecting Asymmetric Conjugate Additions of α-Alkyl-α-cyanoacetates to Acetylenic Esters (Collaboration)
44.	2006	Article	Pattern-based Discrimination of Enantiomeric and Structurally Similar Amino Acids: An Optical Mimic of the Mammalian Taste Response (Collaboration)
45.	2005	Article	Convenient Preparation of Highly Active Phase-transfer Catalyst for Catalytic Asymmetric Synthesis of α-Alkyl- and α,α-Dialkyl-α-amino Acids: Application to the Short Asymmetric Synthesis of BIRT-377 (Collaboration)
46.	2005	Article	Dramatic Rate Enhancement of Asymmetric Phase-transfer-catalyzed Alkylations (Collaboration)
47.	2005	Article	Powerful Chiral Phase-transfer Catalysts for the Asymmetric Synthesis of α-Alkyl- and α,α-Dialkyl-α-amino Acids (Collaboration)
48.	2004	Article	Novel Synthetic Route to Octasubstituted Naphthalenes from Four Alkynes and One Olefin Unit via Zirconacyclopentadienes and 1,2-Diiodo-3,4,5,6-tetraalkylbenzene (Collaboration)
49.	2004	Article	Substituent Effect on Regioselectivity in Oxygenation of Multisubstituted Acenes (Collaboration)
50.	2003	Article	Ortho-metalation of Aromatic Ethers by Yttrium Alkyl Complexes That Contain a Linked Amido-cyclopentadienyl Ligand (Collaboration)
51.	2002	Article	Coupling Reaction of Zirconacyclopentadienes with Dihalonaphthalenes and Dihalopyridines: A New Procedure for the Preparation of Substituted Anthracenes, Quinolines, and Isoquinolines (Collaboration)
52.	2002	Article	Metalation of Aromatic Heterocycles by Yttrium Alkyl Complexes That Contain a Linked Amido-cyclopetadienyl Ligand: Synthesis, Structure and Lewis Base Adduct Formation (Collaboration)
53.	2002	Article	Unusual Conformational Isomer of 9,10-Dihydro-1,2,3,4,5,6,7,8-octapropylanthracene in Solid State (Collaboration)
54.	2001	Article	Aromatization of Highly Alkyl-substituted Dihydroanthracenes Using n-BuLi/TMEDA/MeI (Collaboration)
55.	2000	Article	Straightforward Method for Synthesis of Highly Alkyl-substituted Naphthacene and Pentacene Derivatives by Homologation (Collaboration)
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Invited Lectures

1.	2007	Functional Compounds Prepared with Organometallic Chemistry (Hokkaido)
2.	2015	Intramolecular cyclization using a π-deficient 1,3,5-triazine (Guangdong, China)